Aromatic diamidine compound that binds to kinetoplast DNA (kDNA) minor groove of trypanosomes and Babesia, disrupting DNA replication and transcription. Also inhibits aerobic glycolysis and delta-aminolevulinic acid synthetase in protozoa.
At a glance
Class
Antiprotozoal (Aromatic Diamidine)
Storage
Store at room temperature; reconstituted solution use immediately
Dosing
Used for Babesia canis infection (large Babesia)
Frequency
Once; may repeat once in 24h
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →Safety
PCV and blood smear post-treatmentNeurological assessmentRenal and hepatic functionClinical response at 24–48h
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →Interactions
No documented interactions.
FAQs
Frequently asked questions
›What is Diminazene?
Diminazene is a antiprotozoal (aromatic diamidine) used in pets. Aromatic diamidine compound that binds to kinetoplast DNA (kDNA) minor groove of trypanosomes and Babesia, disrupting DNA replication and transcription. Also inhibits aerobic glycolysis and delta-aminolevulinic acid synthetase in protozoa.
›What is Diminazene used for in pets?
Diminazene is used in veterinary medicine for: Used for Babesia canis infection (large Babesia); Very limited feline data.
›What is the Diminazene dose for dogs?
For dogs, Diminazene is typically dosed as follows — Used for Babesia canis infection (large Babesia): 3.5–5 mg/kg IM (deep injection) Once; may repeat once in 24h. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
›What is the Diminazene dose for cats?
For cats, Diminazene is typically dosed as follows — Very limited feline data: 2 mg/kg IM Once. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
›Does Diminazene need a prescription?
Yes. Diminazene is a prescription medication and should only be administered under veterinary supervision.
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →References
CDSCO approvals (India) — 1
Each ml contains: Diminazene Diaceturate 70 mg+ Phenazone BP 375 mg + chlorocres
M/s. Crescent Lab · Approved 13.02.2015
For the treatment of: Babesiosis caused by B.bovis, B.bigemina, B.motasi & B.canis. Trypanosomoisis caused by T.congolen
Source: CDSCO Veterinary Drug Approval Registry (1969–2026)
References
The PetCare.AI drug reference is built from 13 authoritative sources cited across 580 drug monographs.
Textbooks & handbooks — 5
- Plumb's Veterinary Drug Handbook
- Withrow & MacEwen's Small Animal Clinical Oncology
- Merck Veterinary Manual
- NRC Nutrient Requirements of Dogs and Cats
- Veterinary Pharmacology and Therapeutics (Riviere & Papich)
Clinical guidelines & consensus — 4
- ASPCA Animal Poison Control Center Guidelines
- AAHA Diabetes Management Guidelines
- ASPCA Poison Control Guidelines
- RECOVER CPR Guidelines
Journals & peer-reviewed studies — 2
- EPIC Study (J Vet Intern Med 2016)
- JVIM FAT CAT Study
Regulatory & approvals — 1
- CDSCO Veterinary Drug Approval Registry (1969–2026)
Databases — 1
- Washington State University VCPL MDR1 Database