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Granisetron

Prescription
5-HT3 Serotonin Receptor Antagonist / Antiemetic
Last reviewed 21 Apr 2026 · PetCare.AI Editorial Team
Species
Dog, Cat
Brands
2 available
Formulations
3

Mechanism of action

Selectively blocks 5-HT3 serotonin receptors in the CTZ and vagal afferents, preventing serotonin-induced nausea and vomiting. More selective and longer-acting than ondansetron.

At a glance

Class
5-HT3 Serotonin Receptor Antagonist / Antiemetic
Schedule
Prescription
Storage
Store at room temperature, protect from light

Dosing

🐕

Dog

Used for chemotherapy-induced nausea
Dose
0.1 mg/kg
Route
IV, Transdermal
Frequency
Once per cycle; patch lasts 5–7 days
🐈

Cat

Limited feline data
Dose
0.1 mg/kg
Route
IV
Frequency
Once pre-chemotherapy
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Formulations

💊

Other — 3

Strength
Strength
Strength

Storage

Store at room temperature, protect from light

Safety

Monitoring parameters

Emesis controlCardiac rhythmElectrolytes
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Interactions

No documented interactions.

Brands

Other markets

Kytril
Sancuso (patch)

FAQs

Frequently asked questions

What is Granisetron?
Granisetron is a 5-ht3 serotonin receptor antagonist / antiemetic used in pets. Selectively blocks 5-HT3 serotonin receptors in the CTZ and vagal afferents, preventing serotonin-induced nausea and vomiting. More selective and longer-acting than ondansetron.
What is Granisetron used for in pets?
Granisetron is used in veterinary medicine for: Used for chemotherapy-induced nausea; Limited feline data.
What is the Granisetron dose for dogs?
For dogs, Granisetron is typically dosed as follows — Used for chemotherapy-induced nausea: 0.1 mg/kg IV/Transdermal Once per cycle; patch lasts 5–7 days. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
What is the Granisetron dose for cats?
For cats, Granisetron is typically dosed as follows — Limited feline data: 0.1 mg/kg IV Once pre-chemotherapy. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
Does Granisetron need a prescription?
Yes. Granisetron is a prescription medication and should only be administered under veterinary supervision.
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

References

References

The PetCare.AI drug reference is built from 13 authoritative sources cited across 580 drug monographs.

Textbooks & handbooks — 5

  • Plumb's Veterinary Drug Handbook
  • Withrow & MacEwen's Small Animal Clinical Oncology
  • Merck Veterinary Manual
  • NRC Nutrient Requirements of Dogs and Cats
  • Veterinary Pharmacology and Therapeutics (Riviere & Papich)

Clinical guidelines & consensus — 4

  • ASPCA Animal Poison Control Center Guidelines
  • AAHA Diabetes Management Guidelines
  • ASPCA Poison Control Guidelines
  • RECOVER CPR Guidelines

Journals & peer-reviewed studies — 2

  • EPIC Study (J Vet Intern Med 2016)
  • JVIM FAT CAT Study

Regulatory & approvals — 1

  • CDSCO Veterinary Drug Approval Registry (1969–2026)

Databases — 1

  • Washington State University VCPL MDR1 Database

Related medicines

Other medicines in the same class (5-HT3 Serotonin Receptor Antagonist / Antiemetic).

Dolasetron
Rx
Selectively antagonizes 5-HT3 serotonin receptors in the chemoreceptor trigger zone (CTZ) and peripheral vagal nerve terminals in the GI tract, preventing serotonin-induced nausea and vomiting.
dogcat
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