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Spinosad

Prescription
Spinosyn Insecticide
Last reviewed 21 Apr 2026 · PetCare.AI Editorial Team
Species
Dog, Cat
Brands
2 available
Formulations
1

Mechanism of action

Derived from Saccharopolyspora spinosa fermentation. Activates nicotinic acetylcholine receptors at a unique site, causing involuntary muscle contractions, paralysis, and death of fleas. Also activates GABA receptors at high concentrations.

At a glance

Class
Spinosyn Insecticide
Schedule
Prescription
Storage
Store at room temperature below 30°C

Dosing

🐕

Dog

FDA-approved oral flea treatment
Dose
30 mg/kg
Route
PO
Frequency
Monthly
🐈

Cat

FDA-approved for cats ≥14 weeks and ≥1
Dose
50 mg/kg
Route
PO
Frequency
Monthly
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Formulations

💊

Other — 1

Strength

Storage

Store at room temperature below 30°C

Safety

Monitoring parameters

Flea burden assessmentGI tolerance (first dose)Seizure history
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Interactions

No documented interactions.

Brands

Other markets

Comfortis
Trifexis (with milbemycin)

FAQs

Frequently asked questions

What is Spinosad?
Spinosad is a spinosyn insecticide used in pets. Derived from Saccharopolyspora spinosa fermentation. Activates nicotinic acetylcholine receptors at a unique site, causing involuntary muscle contractions, paralysis, and death of fleas. Also activates GABA receptors at high concentrations.
What is Spinosad used for in pets?
Spinosad is used in veterinary medicine for: FDA-approved oral flea treatment; FDA-approved for cats ≥14 weeks and ≥1.
What is the Spinosad dose for dogs?
For dogs, Spinosad is typically dosed as follows — FDA-approved oral flea treatment: 30 mg/kg PO Monthly. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
What is the Spinosad dose for cats?
For cats, Spinosad is typically dosed as follows — FDA-approved for cats ≥14 weeks and ≥1: 50 mg/kg PO Monthly. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
Does Spinosad need a prescription?
Yes. Spinosad is a prescription medication and should only be administered under veterinary supervision.
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

References

References

The PetCare.AI drug reference is built from 13 authoritative sources cited across 580 drug monographs.

Textbooks & handbooks — 5

  • Plumb's Veterinary Drug Handbook
  • Withrow & MacEwen's Small Animal Clinical Oncology
  • Merck Veterinary Manual
  • NRC Nutrient Requirements of Dogs and Cats
  • Veterinary Pharmacology and Therapeutics (Riviere & Papich)

Clinical guidelines & consensus — 4

  • ASPCA Animal Poison Control Center Guidelines
  • AAHA Diabetes Management Guidelines
  • ASPCA Poison Control Guidelines
  • RECOVER CPR Guidelines

Journals & peer-reviewed studies — 2

  • EPIC Study (J Vet Intern Med 2016)
  • JVIM FAT CAT Study

Regulatory & approvals — 1

  • CDSCO Veterinary Drug Approval Registry (1969–2026)

Databases — 1

  • Washington State University VCPL MDR1 Database
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