Synthetic phospholipid analog that integrates into the parasite cell membrane, disrupting signal transduction, lipid metabolism, and membrane integrity. Also induces apoptosis-like death in Leishmania amastigotes. The only oral treatment for canine leishmaniosis.
At a glance
Class
Alkylphosphocholine Antiprotozoal
Storage
Store at room temperature below 30°C, protect from moisture
Dosing
Licensed in Europe for canine leishmaniosis (Leishmania infantum)
Off-label for feline leishmaniosis
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →Safety
Leishmania serology/PCR post-treatmentRenal function (BUN, creatinine, urinalysis)Hepatic enzymesClinical improvement (skin, lymph nodes)Body weight
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →Interactions
No documented interactions.
FAQs
Frequently asked questions
›What is Miltefosine?
Miltefosine is a alkylphosphocholine antiprotozoal used in pets. Synthetic phospholipid analog that integrates into the parasite cell membrane, disrupting signal transduction, lipid metabolism, and membrane integrity. Also induces apoptosis-like death in Leishmania amastigotes. The only oral treatment for canine leishmaniosis.
›What is Miltefosine used for in pets?
Miltefosine is used in veterinary medicine for: Licensed in Europe for canine leishmaniosis (Leishmania infantum); Off-label for feline leishmaniosis.
›What is the Miltefosine dose for dogs?
For dogs, Miltefosine is typically dosed as follows — Licensed in Europe for canine leishmaniosis (Leishmania infantum): 2 mg/kg PO q24h x 28 days. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
›What is the Miltefosine dose for cats?
For cats, Miltefosine is typically dosed as follows — Off-label for feline leishmaniosis: 2 mg/kg PO q24h x 28 days. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
›Does Miltefosine need a prescription?
Yes. Miltefosine is a prescription medication and should only be administered under veterinary supervision.
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →References
References
The PetCare.AI drug reference is built from 13 authoritative sources cited across 580 drug monographs.
Textbooks & handbooks — 5
- Plumb's Veterinary Drug Handbook
- Withrow & MacEwen's Small Animal Clinical Oncology
- Merck Veterinary Manual
- NRC Nutrient Requirements of Dogs and Cats
- Veterinary Pharmacology and Therapeutics (Riviere & Papich)
Clinical guidelines & consensus — 4
- ASPCA Animal Poison Control Center Guidelines
- AAHA Diabetes Management Guidelines
- ASPCA Poison Control Guidelines
- RECOVER CPR Guidelines
Journals & peer-reviewed studies — 2
- EPIC Study (J Vet Intern Med 2016)
- JVIM FAT CAT Study
Regulatory & approvals — 1
- CDSCO Veterinary Drug Approval Registry (1969–2026)
Databases — 1
- Washington State University VCPL MDR1 Database