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Isotretinoin

Prescription
Systemic Retinoid (Vitamin A Derivative)
Last reviewed 21 Apr 2026 · PetCare.AI Editorial Team
Species
Dog, Cat
Brands
2 available
Formulations
1

Mechanism of action

13-cis-retinoic acid that normalizes keratinization, reduces sebaceous gland size and sebum production (up to 90% reduction), has anti-inflammatory effects, and modulates immune function. Used for keratinization disorders in dogs.

At a glance

Class
Systemic Retinoid (Vitamin A Derivative)
Schedule
Prescription
Storage
Store at room temperature, protect from light and moisture

Dosing

🐕

Dog

Used for idiopathic sebaceous adenitis, sebaceous gland hyperplasia, and lamella
Dose
1–3 mg/kg
Route
PO
Frequency
q24h
🐈

Cat

Very limited feline data
Dose
Route
PO
Frequency
N/A
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Formulations

💊

Other — 1

Strength

Storage

Store at room temperature, protect from light and moisture

Safety

Monitoring parameters

Schirmer tear test baseline and monthly (KCS)Hepatic enzymes q4–8 weeksTriglycerides and cholesterolPregnancy prevention
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Interactions

No documented interactions.

Brands

Other markets

Accutane
Absorica

FAQs

Frequently asked questions

What is Isotretinoin?
Isotretinoin is a systemic retinoid (vitamin a derivative) used in pets. 13-cis-retinoic acid that normalizes keratinization, reduces sebaceous gland size and sebum production (up to 90% reduction), has anti-inflammatory effects, and modulates immune function. Used for keratinization disorders in dogs.
What is Isotretinoin used for in pets?
Isotretinoin is used in veterinary medicine for: Used for idiopathic sebaceous adenitis, sebaceous gland hyperplasia, and lamella; Very limited feline data.
What is the Isotretinoin dose for dogs?
For dogs, Isotretinoin is typically dosed as follows — Used for idiopathic sebaceous adenitis, sebaceous gland hyperplasia, and lamella: 1–3 mg/kg PO q24h. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
What is the Isotretinoin dose for cats?
For cats, Isotretinoin is typically dosed as follows — Very limited feline data: undefined undefined PO N/A. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
Does Isotretinoin need a prescription?
Yes. Isotretinoin is a prescription medication and should only be administered under veterinary supervision.
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

References

References

The PetCare.AI drug reference is built from 13 authoritative sources cited across 580 drug monographs.

Textbooks & handbooks — 5

  • Plumb's Veterinary Drug Handbook
  • Withrow & MacEwen's Small Animal Clinical Oncology
  • Merck Veterinary Manual
  • NRC Nutrient Requirements of Dogs and Cats
  • Veterinary Pharmacology and Therapeutics (Riviere & Papich)

Clinical guidelines & consensus — 4

  • ASPCA Animal Poison Control Center Guidelines
  • AAHA Diabetes Management Guidelines
  • ASPCA Poison Control Guidelines
  • RECOVER CPR Guidelines

Journals & peer-reviewed studies — 2

  • EPIC Study (J Vet Intern Med 2016)
  • JVIM FAT CAT Study

Regulatory & approvals — 1

  • CDSCO Veterinary Drug Approval Registry (1969–2026)

Databases — 1

  • Washington State University VCPL MDR1 Database
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