Partial agonist at the benzodiazepine binding site of GABA-A receptors, with lower intrinsic efficacy than full benzodiazepines (less sedation, less tolerance, less dependence). Also weakly inhibits voltage-gated calcium channels.
At a glance
Class
Low-Affinity Partial Benzodiazepine Agonist / Anticonvulsant
Storage
Store at room temperature below 30°C
Dosing
Licensed for canine idiopathic epilepsy in EU (not FDA-approved in USA)
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →Safety
Seizure frequency diaryBody weight (polyphagia risk)Hepatic enzymes with prolonged use
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →Interactions
No documented interactions.
FAQs
Frequently asked questions
›What is Imepitoin?
Imepitoin is a low-affinity partial benzodiazepine agonist / anticonvulsant used in pets. Partial agonist at the benzodiazepine binding site of GABA-A receptors, with lower intrinsic efficacy than full benzodiazepines (less sedation, less tolerance, less dependence). Also weakly inhibits voltage-gated calcium channels.
›What is Imepitoin used for in pets?
Imepitoin is used in veterinary medicine for: Licensed for canine idiopathic epilepsy in EU (not FDA-approved in USA); Not licensed for cats.
›What is the Imepitoin dose for dogs?
For dogs, Imepitoin is typically dosed as follows — Licensed for canine idiopathic epilepsy in EU (not FDA-approved in USA): 10–30 mg/kg PO q12h. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
›What is the Imepitoin dose for cats?
For cats, Imepitoin is typically dosed as follows — Not licensed for cats: undefined undefined PO N/A. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
›Does Imepitoin need a prescription?
Yes. Imepitoin is a prescription medication and should only be administered under veterinary supervision.
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet.
Find a vet near you →References
References
The PetCare.AI drug reference is built from 13 authoritative sources cited across 580 drug monographs.
Textbooks & handbooks — 5
- Plumb's Veterinary Drug Handbook
- Withrow & MacEwen's Small Animal Clinical Oncology
- Merck Veterinary Manual
- NRC Nutrient Requirements of Dogs and Cats
- Veterinary Pharmacology and Therapeutics (Riviere & Papich)
Clinical guidelines & consensus — 4
- ASPCA Animal Poison Control Center Guidelines
- AAHA Diabetes Management Guidelines
- ASPCA Poison Control Guidelines
- RECOVER CPR Guidelines
Journals & peer-reviewed studies — 2
- EPIC Study (J Vet Intern Med 2016)
- JVIM FAT CAT Study
Regulatory & approvals — 1
- CDSCO Veterinary Drug Approval Registry (1969–2026)
Databases — 1
- Washington State University VCPL MDR1 Database