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Fluorouracil (5-FU)

Prescription
Antimetabolite (Chemotherapy)
Last reviewed 21 Apr 2026 · PetCare.AI Editorial Team
Species
Dog, Cat
Brands
2 available
Formulations
2

Mechanism of action

Pyrimidine analog converted to active metabolites that inhibit thymidylate synthase (blocking DNA synthesis) and incorporate into RNA (disrupting RNA processing). S-phase specific.

At a glance

Class
Antimetabolite (Chemotherapy)
Schedule
Prescription (Chemotherapy)
Storage
Store at room temperature; protect from light; chemotherapy precautions; KEEP AWAY FROM CATS

Dosing

🐕

Dog

Used for various carcinomas
Dose
150 mg/m²
Route
IV
Frequency
Weekly or per protocol
🐈

Cat

NEVER use 5-FU in cats — even small topical exposure causes fatal neurotoxicity
Dose
Route
N, A
Frequency
N/A
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Formulations

💊

Other — 2

Strength
Strength

Storage

Store at room temperature; protect from light; chemotherapy precautions; KEEP AWAY FROM CATS

Safety

Monitoring parameters

CBC at nadirGI toleranceNeurological statusEnsure NO cat contact with treated dog or excreta
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Interactions

No documented interactions.

Brands

Other markets

Efudex
Adrucil

FAQs

Frequently asked questions

What is Fluorouracil (5-FU)?
Fluorouracil (5-FU) is a antimetabolite (chemotherapy) used in pets. Pyrimidine analog converted to active metabolites that inhibit thymidylate synthase (blocking DNA synthesis) and incorporate into RNA (disrupting RNA processing). S-phase specific.
What is Fluorouracil (5-FU) used for in pets?
Fluorouracil (5-FU) is used in veterinary medicine for: Used for various carcinomas; NEVER use 5-FU in cats — even small topical exposure causes fatal neurotoxicity .
What is the Fluorouracil (5-FU) dose for dogs?
For dogs, Fluorouracil (5-FU) is typically dosed as follows — Used for various carcinomas: 150 mg/m² IV Weekly or per protocol. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
What is the Fluorouracil (5-FU) dose for cats?
For cats, Fluorouracil (5-FU) is typically dosed as follows — NEVER use 5-FU in cats — even small topical exposure causes fatal neurotoxicity : undefined undefined N/A N/A. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
Does Fluorouracil (5-FU) need a prescription?
Yes. Fluorouracil (5-FU) is a prescription medication and should only be administered under veterinary supervision.
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

References

References

The PetCare.AI drug reference is built from 13 authoritative sources cited across 580 drug monographs.

Textbooks & handbooks — 5

  • Plumb's Veterinary Drug Handbook
  • Withrow & MacEwen's Small Animal Clinical Oncology
  • Merck Veterinary Manual
  • NRC Nutrient Requirements of Dogs and Cats
  • Veterinary Pharmacology and Therapeutics (Riviere & Papich)

Clinical guidelines & consensus — 4

  • ASPCA Animal Poison Control Center Guidelines
  • AAHA Diabetes Management Guidelines
  • ASPCA Poison Control Guidelines
  • RECOVER CPR Guidelines

Journals & peer-reviewed studies — 2

  • EPIC Study (J Vet Intern Med 2016)
  • JVIM FAT CAT Study

Regulatory & approvals — 1

  • CDSCO Veterinary Drug Approval Registry (1969–2026)

Databases — 1

  • Washington State University VCPL MDR1 Database

Related medicines

Other medicines in the same class (Antimetabolite).

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