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Diphenoxylate/Atropine

Antidiarrheal Opioid Combination
Last reviewed 21 Apr 2026 · PetCare.AI Editorial Team
Species
Dog, Cat
Brands
1 available
Formulations
2

Mechanism of action

Diphenoxylate activates mu-opioid receptors in the GI tract, reducing peristalsis and increasing transit time. Atropine added in sub-therapeutic doses to discourage abuse.

At a glance

Class
Antidiarrheal Opioid Combination
Schedule
Controlled Substance
Storage
Store at room temperature, protect from light

Dosing

🐕

Dog

Used for non-infectious diarrhea only
Dose
0.1–0.2 mg/kg
Route
PO
Frequency
q8–12h
🐈

Cat

Cats more sensitive to opioid effects
Dose
0.05–0.1 mg/kg
Route
PO
Frequency
q12h
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Formulations

💊

Other — 2

Strength
Strength

Storage

Store at room temperature, protect from light

Safety

Monitoring parameters

Stool frequencyResolution within 48hHydration status
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

Interactions

No documented interactions.

Brands

Other markets

Lomotil

FAQs

Frequently asked questions

What is Diphenoxylate/Atropine?
Diphenoxylate/Atropine is a antidiarrheal opioid combination used in pets. Diphenoxylate activates mu-opioid receptors in the GI tract, reducing peristalsis and increasing transit time. Atropine added in sub-therapeutic doses to discourage abuse.
What is Diphenoxylate/Atropine used for in pets?
Diphenoxylate/Atropine is used in veterinary medicine for: Used for non-infectious diarrhea only; Cats more sensitive to opioid effects.
What is the Diphenoxylate/Atropine dose for dogs?
For dogs, Diphenoxylate/Atropine is typically dosed as follows — Used for non-infectious diarrhea only: 0.1–0.2 mg/kg PO q8–12h. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
What is the Diphenoxylate/Atropine dose for cats?
For cats, Diphenoxylate/Atropine is typically dosed as follows — Cats more sensitive to opioid effects: 0.05–0.1 mg/kg PO q12h. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
Does Diphenoxylate/Atropine need a prescription?
Diphenoxylate/Atropine is available over the counter. Even so, you should consult your veterinarian before giving any medication to your pet.
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →

References

References

The PetCare.AI drug reference is built from 13 authoritative sources cited across 580 drug monographs.

Textbooks & handbooks — 5

  • Plumb's Veterinary Drug Handbook
  • Withrow & MacEwen's Small Animal Clinical Oncology
  • Merck Veterinary Manual
  • NRC Nutrient Requirements of Dogs and Cats
  • Veterinary Pharmacology and Therapeutics (Riviere & Papich)

Clinical guidelines & consensus — 4

  • ASPCA Animal Poison Control Center Guidelines
  • AAHA Diabetes Management Guidelines
  • ASPCA Poison Control Guidelines
  • RECOVER CPR Guidelines

Journals & peer-reviewed studies — 2

  • EPIC Study (J Vet Intern Med 2016)
  • JVIM FAT CAT Study

Regulatory & approvals — 1

  • CDSCO Veterinary Drug Approval Registry (1969–2026)

Databases — 1

  • Washington State University VCPL MDR1 Database
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