Home/Medicines/Bupivacaine Liposome
All medicines

Bupivacaine Liposome

Prescription
Extended-Release Local Anesthetic
Last reviewed 21 Apr 2026 · PetCare.AI Editorial Team
Species
Dog, Cat
Brands
1 available
Formulations
1

Mechanism of action

Liposomal encapsulation of bupivacaine that provides sustained drug release over 72h from a single injection, blocking voltage-gated sodium channels and preventing pain signal transmission for significantly longer than standard bupivacaine (4–8h).

At a glance

Class
Extended-Release Local Anesthetic
Schedule
Prescription
Storage
Refrigerate 2–8°C; can be at room temperature up to 30 days; do not freeze; gently invert to mix — do not shake

Dosing

🐕

Dog

FDA-approved for post-operative analgesia at surgical sites in dogs
Dose
5.3 mg/kg
Route
PO
Frequency
Once per surgical site
🐈

Cat

FDA-approved for cats (onychectomy/declaw — where still performed)
Dose
5.3 mg/kg
Route
Local infiltration
Frequency
Once

Formulations

💊

Other — 1

Strength

Storage

Refrigerate 2–8°C; can be at room temperature up to 30 days; do not freeze; gently invert to mix — do not shake

Safety

Monitoring parameters

Pain scores for 72h post-surgerySurgical site healingSigns of systemic toxicity

Interactions

No documented interactions.

Brands

Other markets

Nocita

FAQs

Frequently asked questions

What is Bupivacaine Liposome?
Bupivacaine Liposome is a extended-release local anesthetic used in pets. Liposomal encapsulation of bupivacaine that provides sustained drug release over 72h from a single injection, blocking voltage-gated sodium channels and preventing pain signal transmission for significantly longer than standard bupivacaine (4–8h).
What is Bupivacaine Liposome used for in pets?
Bupivacaine Liposome is used in veterinary medicine for: FDA-approved for post-operative analgesia at surgical sites in dogs; FDA-approved for cats (onychectomy/declaw — where still performed).
What is the Bupivacaine Liposome dose for dogs?
For dogs, Bupivacaine Liposome is typically dosed as follows — FDA-approved for post-operative analgesia at surgical sites in dogs: 5.3 mg/kg PO Once per surgical site. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
What is the Bupivacaine Liposome dose for cats?
For cats, Bupivacaine Liposome is typically dosed as follows — FDA-approved for cats (onychectomy/declaw — where still performed): 5.3 mg/kg Local infiltration Once. Always consult your veterinarian for a dose tailored to your pet's weight, age, and condition.
Does Bupivacaine Liposome need a prescription?
Yes. Bupivacaine Liposome is a prescription medication and should only be administered under veterinary supervision.

References

References

Textbooks & handbooks

  • Plumb, D.C. Plumb's Veterinary Drug Handbook. 10th ed., Wiley-Blackwell, 2023.
  • Vail, D.M., Thamm, D.H., & Liptak, J.M. (eds.). Withrow & MacEwen's Small Animal Clinical Oncology. 6th ed., Saunders/Elsevier, 2020.
  • Riviere, J.E., & Papich, M.G. (eds.). Veterinary Pharmacology and Therapeutics. 10th ed., Wiley-Blackwell, 2018.
  • National Research Council. Nutrient Requirements of Dogs and Cats. National Academies Press, Washington DC, 2006.
  • The Merck Veterinary Manual. Merck & Co., Online edition. https://www.merckvetmanual.com/

Clinical guidelines & consensus

  • Fletcher, D.J., Boller, M., Brainard, B.M., et al. "RECOVER Evidence and Knowledge Gap Analysis on Veterinary CPR." Journal of Veterinary Emergency and Critical Care, 2012;22(S1):S102–S131.
  • American Animal Hospital Association. 2018 AAHA Diabetes Management Guidelines for Dogs and Cats. AAHA Press.

Journals & peer-reviewed studies

  • Hogan, D.F., Fox, P.R., Jacob, K., et al. "Secondary prevention of cardiogenic arterial thromboembolism in the cat: The FAT CAT study." Journal of Veterinary Cardiology, 2015;17(Suppl 1):S306–S317.
  • Boswood, A., Häggström, J., Gordon, S.G., et al. "Effect of Pimobendan in Dogs with Preclinical Myxomatous Mitral Valve Disease and Cardiomegaly: The EPIC Study — A Randomized Clinical Trial." Journal of Veterinary Internal Medicine, 2016;30(6):1765–1779.
  • ASPCA Animal Poison Control Center. Toxicology and Poison Management Guidelines. American Society for the Prevention of Cruelty to Animals. https://www.aspca.org/pet-care/animal-poison-control

Regulatory & approvals

  • Central Drugs Standard Control Organisation (CDSCO), Government of India. Veterinary Drug Approval Registry, 1969–2026. Directorate General of Health Services. https://cdsco.gov.in/

Databases

  • Washington State University, College of Veterinary Medicine. Veterinary Clinical Pharmacology Laboratory (VCPL) — MDR1 Multidrug Sensitivity Database. https://vcpl.vetmed.wsu.edu/
Educational reference only
This information is provided for educational purposes and is not a substitute for professional veterinary advice, diagnosis, or treatment. Always consult a qualified veterinarian before administering any medication to your pet. Find a vet near you →